Discovery:
Discovery:
developing synthetic macrocycles and other creative small molecule solutionsRead more...

								Expertise:
Expertise:
expanding the boundaries of traditional therapeuticsRead more...

								Pipeline:
Pipeline:
advancing small molecule therapies for patients with cancer and other serious diseasesRead more...

								Partnering:
Partnering:
demonstrating success against challenging disease targets in collaboration with global partnersRead more...

Ensemble is focused on the discovery and development of breakthrough small molecule therapies for patients with cancer and other serious diseases. We are aggressively applying our proprietary drug discovery platform to go beyond the boundaries of traditional therapeutics by developing novel small molecules against challenging disease targets.

Discovery Platform
Designing and optimizing innovative small molecules
Designing and optimizing innovative small molecules
Pipeline
Designing and optimizing innovative small molecules
Developing immune checkpoint and ubiquitin proteasome inhibitors
Ensemble is committed to providing safer and more effective treatments for patients
Ensemble is committed to providing safer and more effective treatments for patients
Spotlight
XIAP linear and macrocyle overlap 166 x 166
Feb 5, 2016
How Beyond ‘Rule of 5’ Drugs Bind to Proteins
4AQK PD1_PD-L1 protein strcuture_166x166
Jan 13, 2016
New PD-1 Protein Structure Will Aid Macrocycle Inhibitor Design
spotlight-poster
Sep 25, 2015
Ensemble Scientist Awarded First Place at the 2015 Discovery on Target Conference Poster Competition